| Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus M Bassetto, T De Burghgraeve, L Delang, A Massarotti, A Coluccia, ... Antiviral research 98 (1), 12-18, 2013 | 114 | 2013 |
| Synthesis and Biological Evaluation of 2-(Alkoxycarbonyl)-3-Anilinobenzo[b]thiophenes and Thieno[2,3-b]pyridines as New Potent Anticancer Agents R Romagnoli, PG Baraldi, M Kimatrai Salvador, D Preti, ... Journal of medicinal chemistry 56 (6), 2606-2618, 2013 | 110 | 2013 |
| Polyfluorinated groups in medicinal chemistry M Bassetto, S Ferla, F Pertusati Future Medicinal Chemistry 7 (4), 527-546, 2015 | 108 | 2015 |
| Synthesis and biological evaluation of 2-substituted-4-(3′, 4′, 5′-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents R Romagnoli, PG Baraldi, MK Salvador, ME Camacho, D Preti, MA Tabrizi, ... Bioorganic & medicinal chemistry 20 (24), 7083-7094, 2012 | 77 | 2012 |
| Design and synthesis of novel bicalutamide and enzalutamide derivatives as antiproliferative agents for the treatment of prostate cancer M Bassetto, S Ferla, F Pertusati, S Kandil, AD Westwell, A Brancale, ... European Journal of Medicinal Chemistry 118, 230-243, 2016 | 70 | 2016 |
| Concise Synthesis and Biological Evaluation of 2-Aroyl-5-Amino Benzo[b]thiophene Derivatives As a Novel Class of Potent Antimitotic Agents R Romagnoli, PG Baraldi, C Lopez-Cara, D Preti, M Aghazadeh Tabrizi, ... Journal of medicinal chemistry 56 (22), 9296-9309, 2013 | 65 | 2013 |
| Design, synthesis and biological evaluation of 3, 5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents R Romagnoli, PG Baraldi, C Lopez-Cara, MK Salvador, D Preti, ... Bioorganic & medicinal chemistry 22 (18), 5097-5109, 2014 | 45 | 2014 |
| Computer-aided identification, synthesis and evaluation of substituted thienopyrimidines as novel inhibitors of HCV replication M Bassetto, P Leyssen, J Neyts, MM Yerukhimovich, DN Frick, A Brancale European Journal of Medicinal Chemistry 123, 31-47, 2016 | 33 | 2016 |
| SARS-CoV-2 Virus− Host interaction: currently available structures and implications of variant emergence on infectivity and immune response L Queirós-Reis, P Gomes da Silva, J Gonçalves, A Brancale, M Bassetto, ... International journal of molecular sciences 22 (19), 10836, 2021 | 32 | 2021 |
| In silico screening for human norovirus antivirals reveals a novel non-nucleoside inhibitor of the viral polymerase S Ferla, NE Netzler, S Ferla, S Veronese, DE Tuipulotu, S Guccione, ... Scientific reports 8 (1), 4129, 2018 | 30 | 2018 |
| Diketo acids inhibit the cap-snatching endonuclease of several Bunyavirales Y Fernández-García, S Ter Horst, M Bassetto, A Brancale, J Neyts, ... Antiviral Research 183, 104947, 2020 | 29 | 2020 |
| Antivirals in medical biodefense JJ Bugert, F Hucke, P Zanetta, M Bassetto, A Brancale Virus Genes 56, 150-167, 2020 | 29 | 2020 |
| Targeting the viral polymerase of diarrhea-causing viruses as a strategy to develop a single broad-spectrum antiviral therapy M Bassetto, J Van Dycke, J Neyts, A Brancale, J Rocha-Pereira Viruses 11 (2), 173, 2019 | 27 | 2019 |
| Therapeutically targeting guanylate cyclase‐C: computational modeling of plecanatide, a uroguanylin analog A Brancale, K Shailubhai, S Ferla, A Ricci, M Bassetto, GS Jacob Pharmacology Research & Perspectives 5 (2), e00295, 2017 | 27 | 2017 |
| In silico identification, design and synthesis of novel piperazine-based antiviral agents targeting the hepatitis C virus helicase M Bassetto, P Leyssen, J Neyts, MM Yerukhimovich, DN Frick, ... European journal of medicinal chemistry 125, 1115-1131, 2017 | 26 | 2017 |
| Targeting the complement serine protease MASP-2 as a therapeutic strategy for coronavirus infections BM Flude, G Nannetti, P Mitchell, N Compton, C Richards, M Heurich, ... Viruses 13 (2), 312, 2021 | 24 | 2021 |
| Rational design of highly potent broad-spectrum enterovirus inhibitors targeting the nonstructural protein 2C L Bauer, R Manganaro, B Zonsics, DL Hurdiss, M Zwaagstra, T Donselaar, ... PLoS Biology 18 (11), e3000904, 2020 | 24 | 2020 |
| Rational modifications on a benzylidene-acrylohydrazide antiviral scaffold, synthesis and evaluation of bioactivity against Chikungunya virus G Giancotti, M Cancellieri, A Balboni, M Giustiniano, E Novellino, ... European Journal of Medicinal Chemistry 149, 56-68, 2018 | 24 | 2018 |
| A new series of bicalutamide, enzalutamide and enobosarm derivatives carrying pentafluorosulfanyl (SF5) and pentafluoroethyl (C2F5) substituents: Improved antiproliferative … F Pertusati, S Ferla, M Bassetto, A Brancale, S Khandil, AD Westwell, ... European Journal of Medicinal Chemistry 180, 1-14, 2019 | 22 | 2019 |
| Design, synthesis and evaluation against Chikungunya virus of novel small-molecule antiviral agents R Tardugno, G Giancotti, T De Burghgraeve, L Delang, J Neyts, ... Bioorganic & Medicinal Chemistry 26 (4), 869-874, 2018 | 22 | 2018 |
