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Adegoke Adeniji
Adegoke Adeniji
South University School of Pharmacy
Verified email at southuniversity.edu
Title
Cited by
Cited by
Year
AKR1C3 as a target in castrate resistant prostate cancer
AO Adeniji, M Chen, TM Penning
The Journal of steroid biochemistry and molecular biology 137, 136-149, 2013
1462013
Development of Potent and Selective Inhibitors of Aldo–Keto Reductase 1C3 (Type 5 17β-Hydroxysteroid Dehydrogenase) Based on N-Phenyl-Aminobenzoates …
AO Adeniji, BM Twenter, MC Byrns, Y Jin, M Chen, JD Winkler, ...
Journal of medicinal chemistry 55 (5), 2311-2323, 2012
1162012
Development of potent and selective indomethacin analogues for the inhibition of AKR1C3 (type 5 17β-hydroxysteroid dehydrogenase/prostaglandin F synthase) in castrate-resistant …
AJ Liedtke, AO Adeniji, M Chen, MC Byrns, Y Jin, DW Christianson, ...
Journal of medicinal chemistry 56 (6), 2429-2446, 2013
1052013
Discovery of substituted 3-(phenylamino) benzoic acids as potent and selective inhibitors of type 5 17β-hydroxysteroid dehydrogenase (AKR1C3)
AO Adeniji, BM Twenter, MC Byrns, Y Jin, JD Winkler, TM Penning
Bioorganic & medicinal chemistry letters 21 (5), 1464-1468, 2011
592011
Crystal structures of AKR1C3 containing an N-(aryl) amino-benzoate inhibitor and a bifunctional AKR1C3 inhibitor and androgen receptor antagonist. Therapeutic leads for …
M Chen, AO Adeniji, BM Twenter, JD Winkler, DW Christianson, ...
Bioorganic & medicinal chemistry letters 22 (10), 3492-3497, 2012
552012
Discovery of (R)-2-(6-Methoxynaphthalen-2-yl)butanoic Acid as a Potent and Selective Aldo-keto Reductase 1C3 Inhibitor
A Adeniji, MJ Uddin, T Zang, D Tamae, P Wangtrakuldee, LJ Marnett, ...
Journal of medicinal chemistry 59 (16), 7431-7444, 2016
412016
Selective inhibitors of aldo-keto reductases AKR1C1 and AKR1C3 discovered by virtual screening of a fragment library
P Brožič, S Turk, AO Adeniji, J Konc, D Janežič, TM Penning, ...
Journal of medicinal chemistry 55 (17), 7417-7424, 2012
272012
A 3-(4-nitronaphthen-1-yl) amino-benzoate analog as a bifunctional AKR1C3 inhibitor and AR antagonist: Head to head comparison with other advanced AKR1C3 targeted therapeutics
P Wangtrakuldee, AO Adeniji, T Zang, L Duan, B Khatri, BM Twenter, ...
The Journal of steroid biochemistry and molecular biology 192, 105283, 2019
202019
N-Benzoyl anthranilic acid derivatives as selective inhibitors of aldo–keto reductase AKR1C3
M Sinreih, I Sosič, N Beranič, S Turk, AO Adeniji, TM Penning, TL Rižner, ...
Bioorganic & medicinal chemistry letters 22 (18), 5948-5951, 2012
202012
Amyloid β hypothesis in the development of therapeutic agents for Alzheimer’s disease
AO Adeniji, PW Adams, VV Mody
Drug Discovery Approaches for the Treatment of Neurodegenerative Disorders …, 2017
132017
Colorimetric assay of naproxen tablets by derivatization using 4-carboxyl-2, 6-dinitrobenzene diazonium ion
SO Idowu, OA Adegoke, AO Adeniji, AA Olaniyi
East and Central African Journal of pharmaceutical sciences 12 (1), 2009
112009
Syntheses and In-Vitro Evaluation of Novel Adamantane Based γ-Secretase Inhibitors
A O Adeniji, R M Wells, A Adejare
Current medicinal chemistry 19 (15), 2458-2471, 2012
82012
Indomethacin analogs for the treatment of castrate-resistant prostate cancer
LJ Marnett, AJ Liedtke, TM Penning, AO Adeniji, MC Byrns
US Patent 9,346,803, 2016
52016
Bifunctional AKR1C3 inhibitors/androgen receptor modulators and methods of use thereof
TM Penning, AO Adeniji, MC Burns, J Winkler, B Twenter
US Patent 9,271,961, 2016
32016
Indomethacin analogs for the treatment of castrate-resistant prostate cancer
LJ Marnett, AJ Liedtke, TM Penning, AO Adeniji, MC Byrns
US Patent 10,398,678, 2019
22019
Crystal structures of human 17β-hydroxysteroid dehydrogenase Type 5 (AKR1C3) in complex with N-phenylanthranilic acid and indomethacin-based selective inhibitors
M Chen, AO Adeniji, BM Twenter, AJ Liedtke, JD Winkler, LJ Marnett, ...
Endocrine Reviews 33 (03_MeetingAbstracts), SAT-536, 2012
22012
Development of potent and selective indomethacin analogs for the inhibition of AKR1C3 in castrate-resistant prostate cancer
AO Adeniji, A Liedtke, MC Byrns, Y Jin, LJ Marnett, TM Penning
Endocr. Rev 33, 2012
22012
Indomethacin analogs for the treatment of castrate-resistant prostate cancer
LJ Marnett, AJ Liedtke, TM Penning, AO Adeniji, MC Byrns
US Patent 11,738,004, 2023
12023
Indomethacin analogs for the treatment of castrate-resistant prostate cancer
LJ Marnett, AJ Liedtke, TM Penning, AO Adeniji, MC Byrns
US Patent App. 16/530,907, 2019
12019
Structure activity relationship (SAR) studies of a novel γ-secretase inhibitor
A Adeniji
University of the Sciences in Philadelphia, 2010
12010
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