C7-Derivatization of C3-Alkylindoles Including Tryptophans and Tryptamines RP Loach, OS Fenton, K Amaike, DS Siegel, E Ozkal, M Movassaghi The Journal of organic chemistry 79 (22), 11254-11263, 2014 | 114 | 2014 |
Employing Photoredox Catalysis for DNA‐Encoded Chemistry: Decarboxylative Alkylation of α‐Amino Acids DK Kölmel, RP Loach, T Knauber, ME Flanagan ChemMedChem 13 (20), 2159-2165, 2018 | 97 | 2018 |
Employing Photoredox Catalysis for DNA‐Encoded Chemistry: Decarboxylative Alkylation of α‐Amino Acids DK Kölmel, RP Loach, T Knauber, ME Flanagan ChemMedChem 13 (20), 2159-2165, 2018 | 97 | 2018 |
General, regiodefined access to alpha-substituted butenolides through metal-halogen exchange of 3-bromo-2-silyloxyfurans. Efficient synthesis of an anti-inflammatory gorgonian … J Boukouvalas, RP Loach The Journal of organic chemistry 73 (20), 8109-8112, 2008 | 90 | 2008 |
On-DNA Decarboxylative Arylation: The Merger of Photoredox with Nickel Catalysis in Water DK Kölmel, J Meng, MH Tsai, J Que, RP Loach, T Knauber, J Wan, ... ACS Combinatorial Science, 2019 | 79 | 2019 |
Concise Total Synthesis of (+)-Asperazine, (+)-Pestalazine A, and (+)-iso-Pestalazine A. Structure Revision of (+)-Pestalazine A RP Loach, OS Fenton, M Movassaghi Journal of the American Chemical Society 138 (3), 1057-1064, 2016 | 61 | 2016 |
Unified route to asymmetrically substituted butenolide, maleic anhydride, and maleimide constituents of Antrodia camphorata J Boukouvalas, V Albert, RP Loach, R Lafleur-Lambert Tetrahedron 68 (47), 9592-9597, 2012 | 28 | 2012 |
Oxidative rearrangement of 2-furylcarbamates with dimethyldioxirane: a high-yielding preparation of 5-hydroxypyrrol-2 (5H)-ones J Boukouvalas, RP Loach, E Ouellet Tetrahedron letters 52 (39), 5047-5050, 2011 | 25 | 2011 |
Concise total synthesis of (+)-asperazine A and (+)-pestalazine B BM Nelson, RP Loach, S Schiesser, M Movassaghi Organic & biomolecular chemistry 16 (2), 202-207, 2018 | 19 | 2018 |
Concise Total Synthesis of (−)-Auxofuran by a Click Diels–Alder Strategy J Boukouvalas, RP Loach Organic letters 15 (18), 4912-4914, 2013 | 16 | 2013 |
Direct C7 Functionalization of Tryptophan. Synthesis of Methyl (S)‐2‐((tert‐Butoxycarbonyl)amino)‐3‐(7‐(4,4,5,5‐tetramethyl‐1,3,2‐dioxaborolan‐2‐yl)‐1H‐indol … K Amaike, RP Loach, M Movassaghi* 2 Organic Syntheses 92, 373-385, 2003 | 14* | 2003 |
Aminolactone Chiral Modifiers for Heterogeneous Asymmetric Hydrogenation: Corrected Structure of Pantoyl-Naphthylethylamine, in-Situ Hydrogenolysis, and Scanning Tunneling … G Goubert, V Demers-Carpentier, RP Loach, R Lafleur-Lambert, ... ACS Catalysis 3 (12), 2677-2683, 2013 | 13 | 2013 |
α-Chiral amines via thermally promoted deaminative addition of alkylpyridinium salts to sulfinimines KM Baker, A Tallon, RP Loach, OP Bercher, MA Perry, MP Watson Organic letters 23 (20), 7735-7739, 2021 | 11 | 2021 |
Early Clinical Development of Lufotrelvir as a Potential Therapy for COVID-19 C Allais, D Bernhardson, AR Brown, GM Chinigo, JN Desrosiers, ... Organic Process Research & Development, 2023 | 10 | 2023 |
Dimethyldioxirane oxidation of 2-silyloxypyrroles: An efficient regiocontrolled synthesis of 5-hydroxy-3-pyrrolin-2-ones J Boukouvalas, Y Xiao, YX Cheng, RP Loach Synlett 2007 (20), 3198-3200, 2007 | 6 | 2007 |
Expedient Assembly of Bioactive Maleic Anhydrides Using Click Diels–Alder Chemistry J Boukouvalas, C Thibault, RP Loach Synlett 25 (15), 2139-2142, 2014 | 3 | 2014 |
Front Cover: Employing Photoredox Catalysis for DNA‐Encoded Chemistry: Decarboxylative Alkylation of α‐Amino Acids (ChemMedChem 20/2018) DK Kölmel, RP Loach, T Knauber, ME Flanagan ChemMedChem 13 (20), 2132-2132, 2018 | 1 | 2018 |
Total synthesis of gamma-hydroxybutenolide-containing acetogenins R Muddala, R Loach, J Boukouvalas ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 251, 2016 | | 2016 |
C7-derivatization of tryptophans and tryptamines for the synthesis of complex alkaloids R Loach, O Fenton, K Amaike, D Siegel, E Ozkal, M Movassaghi ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 250, 2015 | | 2015 |
C7-Derivatization of Tryptophans and Tryptamines for the Synthesis of Complex Alkaloids MM Richard P. Loach, Owen S. Fenton, Kazuma Amaike, Dustin S. Siegel, Erhan ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 245, 2015 | | 2015 |