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Athanasios Papakyriakou
Athanasios Papakyriakou
Institute of Biosciences and Applications, NCSR "Demokritos"
Verified email at bio.demokritos.gr - Homepage
Title
Cited by
Cited by
Year
Dietary flavonoids in cancer therapy and prevention: substrates and inhibitors of cytochrome P450 CYP1 enzymes
VP Androutsopoulos, A Papakyriakou, D Vourloumis, AM Tsatsakis, ...
Pharmacology & therapeutics 126 (1), 9-20, 2010
2382010
The internal sequence of the peptide-substrate determines its N-terminus trimming by ERAP1
I Evnouchidou, F Momburg, A Papakyriakou, A Chroni, L Leondiadis, ...
PloS one 3 (11), e3658, 2008
1292008
Comparative CYP1A1 and CYP1B1 substrate and inhibitor profile of dietary flavonoids
VP Androutsopoulos, A Papakyriakou, D Vourloumis, DA Spandidos
Bioorganic & medicinal chemistry 19 (9), 2842-2849, 2011
1212011
Probing the S1 specificity pocket of the aminopeptidases that generate antigenic peptides
E Zervoudi, A Papakyriakou, D Georgiadou, I Evnouchidou, A Gajda, ...
Biochemical Journal 435 (2), 411-420, 2011
1162011
Synthesis and biopharmaceutical evaluation of imatinib analogues featuring unusual structural motifs
KC Nicolaou, D Vourloumis, S Totokotsopoulos, A Papakyriakou, ...
ChemMedChem 11 (1), 31-37, 2016
1112016
Mononuclear metal complexes with Piroxicam: Synthesis, structure and biological activity
P Christofis, M Katsarou, A Papakyriakou, Y Sanakis, N Katsaros, ...
Journal of inorganic biochemistry 99 (11), 2197-2210, 2005
1022005
A common single nucleotide polymorphism in endoplasmic reticulum aminopeptidase 2 induces a specificity switch that leads to altered antigen processing
I Evnouchidou, J Birtley, S Seregin, A Papakyriakou, E Zervoudi, ...
The Journal of Immunology 189 (5), 2383-2392, 2012
902012
Anticancer effects of the metabolic products of the resveratrol analogue, DMU-212: structural requirements for potency
VP Androutsopoulos, KC Ruparelia, A Papakyriakou, H Filippakis, ...
European Journal of Medicinal Chemistry 46 (6), 2586-2595, 2011
682011
Effects of polymorphic variation on the mechanism of Endoplasmic Reticulum Aminopeptidase 1
A Stamogiannos, D Koumantou, A Papakyriakou, E Stratikos
Molecular immunology 67 (2), 426-435, 2015
662015
Optimization and structure–activity relationships of phosphinic pseudotripeptide inhibitors of aminopeptidases that generate antigenic peptides
P Kokkala, A Mpakali, FX Mauvais, A Papakyriakou, I Daskalaki, ...
Journal of Medicinal Chemistry 59 (19), 9107-9123, 2016
622016
A new role for Zn (II) aminopeptidases: antigenic peptide generation and destruction
I Evnouchidou, A Papakyriakou, E Stratikos
Current pharmaceutical design 15 (31), 3656-3670, 2009
572009
Pyrrolo[2,3-a]carbazoles as Potential Cyclin Dependent Kinase 1 (CDK1) Inhibitors. Synthesis, Biological Evaluation, and Binding Mode through Docking Simulations
MA Fousteris, A Papakyriakou, A Koutsourea, M Manioudaki, ...
Journal of medicinal chemistry 51 (4), 1048-1052, 2008
512008
Crystal structure of insulin-regulated aminopeptidase with bound substrate analogue provides insight on antigenic epitope precursor recognition and processing
A Mpakali, E Saridakis, K Harlos, Y Zhao, A Papakyriakou, P Kokkala, ...
The Journal of Immunology 195 (6), 2842-2851, 2015
502015
Molecular interaction of α-conotoxin RgIA with the rat α9α10 nicotinic acetylcholine receptor
L Azam, A Papakyriakou, M Zouridakis, P Giastas, SJ Tzartos, ...
Molecular pharmacology 87 (5), 855-864, 2015
482015
Crystal structure of the monomeric extracellular domain of α9 nicotinic receptor subunit in complex with α-conotoxin RgIA: Molecular dynamics insights into RgIA binding to …
M Zouridakis, A Papakyriakou, IA Ivanov, IE Kasheverov, V Tsetlin, ...
Frontiers in pharmacology 10, 436925, 2019
472019
Mechanism for antigenic peptide selection by endoplasmic reticulum aminopeptidase 1
P Giastas, A Mpakali, A Papakyriakou, A Lelis, P Kokkala, M Neu, ...
Proceedings of the National Academy of Sciences 116 (52), 26709-26716, 2019
412019
Ligand-induced conformational change of insulin-regulated aminopeptidase: insights on catalytic mechanism and active site plasticity
A Mpakali, E Saridakis, K Harlos, Y Zhao, P Kokkala, D Georgiadis, ...
Journal of Medicinal Chemistry 60 (7), 2963-2972, 2017
392017
Identification of novel melanin synthesis inhibitors from Crataegus pycnoloba using an in vivo zebrafish phenotypic assay
A Agalou, M Thrapsianiotis, A Angelis, A Papakyriakou, AL Skaltsounis, ...
Frontiers in Pharmacology 9, 328125, 2018
372018
3, 4-diaminobenzoic acid derivatives as inhibitors of the oxytocinase subfamily of M1 aminopeptidases with immune-regulating properties
A Papakyriakou, E Zervoudi, S Tsoukalidou, FX Mauvais, G Sfyroera, ...
Journal of medicinal chemistry 58 (3), 1524-1543, 2015
372015
Editing the immunopeptidome of melanoma cells using a potent inhibitor of endoplasmic reticulum aminopeptidase 1 (ERAP1)
D Koumantou, E Barnea, A Martin-Esteban, Z Maben, A Papakyriakou, ...
Cancer Immunology, Immunotherapy 68, 1245-1261, 2019
362019
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